Profiles of Drug Substances, Excipients, and Related Methodology /

Profiles of Drug Substances, Excipients, and Related Methodology, Volume 49 provides timely and pertinent information on a variety of timely topics, including Physical Profiles of Drug Substances and Excipients; Analytical Profiles of Drug Substances and Excipients; ADME Profiles of Drug Substances...

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Bibliographic Details
Corporate Author: ScienceDirect (Online service)
Other Authors: Al-Majed, Abdulrahman (Editor)
Format: eBook
Language:English
Published: London, England : Academic Press, [2024]
Edition:First edition.
Series:Profiles of drug substances, excipients, and related methodology ; Volume 49.
Subjects:
Online Access:Connect to the full text of this electronic book

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490 1 |a Profiles of Drug Substances, Excipients and Related Methodology Series ;  |v Volume 49 
520 |a Profiles of Drug Substances, Excipients, and Related Methodology, Volume 49 provides timely and pertinent information on a variety of timely topics, including Physical Profiles of Drug Substances and Excipients; Analytical Profiles of Drug Substances and Excipients; ADME Profiles of Drug Substances and Excipients; Methodology Related to the Characterization of Drug Substances and Excipients; and Methods of Chemical Synthesis. In addition, it includes comprehensive profiles of five drug compounds: Deferasirox, Duvelisib, Regorafenib, Ponatinib and Avanafil. Finally, the book contains a chapter on Regulation and Standardization of Herbal Drugs: Current status, Limitation, Challenge's, and Future Prospectives. 
505 0 |a Front Cover -- Series Page -- Title Page -- Copyright -- Contents -- Contributors -- Preface -- Chapter One: Deferasirox: A comprehensive drug profileDeferasirox: A comprehensive drug profile -- 1 Description -- 1.1 History -- 1.2 Nomenclature -- 1.2.1 Systemic chemical name -- 1.2.2 Nonproprietary names -- 1.2.3 Proprietary names -- 1.3 Formulae -- 2 Mode of action -- 3 Pharmacokinetics -- 4 Indications -- 5 Synthesis -- 6 Physical characteristics -- 6.1 Solubility -- 6.2 Dissociation constant -- 6.3 Optical activity -- 6.4 Density -- 6.5 Partition coefficient -- 6.6 Melting behavior -- 6.7 Lattice analysis by X-ray powder diffraction -- 6.8 Thermal analysis -- 6.9 FTIR spectroscopy -- 6.10 NMR spectroscopic analysis -- 7 Methods of analysis -- 7.1 Reversed phase-high performance liquid chromatography (RP-HPLC) method -- 7.2 Liquid chromatography combined with tandem mass spectrometry (LC-MS/MS) methods -- 7.3 Spectrophotometric methods -- 7.4 Fluorescence methods -- Acknowledgment -- References -- Chapter Two: Duvelisib: A comprehensive profile -- 1 Description -- 1.1 Nomenclature -- 1.1.1 Systemic chemical names [1] -- 1.1.2 Nonproprietary names [1] -- 1.2 Formulae -- 1.2.1 Empirical formula -- 1.2.2 Structural formula -- 1.3 Elemental composition -- 1.4 Appearance [2,3] -- 1.5 Physicochemical properties [4,5] -- 2 Uses and applications -- 3 Methods of preparation -- 4 Spectroscopic analysis -- 4.1 Ultraviolet-visible spectroscopy -- 4.2 Fluorescence spectroscopy -- 4.3 Fourier-transform infrared absorption spectroscopy -- 4.4 1H-nuclear magnetic resonance spectrometry -- 4.5 Mass spectrometry -- 5 Thermogravimetric analysis -- 6 Methods of analysis -- 6.1 Compendial method -- 6.2 Spectroscopic methods -- 6.2.1 Ultraviolet-visible spectrophotometry -- 6.2.2 Spectrofluorometry -- 6.3 Chromatographic methods -- 7 Pharmacological properties. 
505 8 |a 7.1 Mechanism of action -- 7.2 Pharmacokinetics -- 8 Dosing information -- 8.1 Dosage forms and administration -- 8.2 Contraindications -- 8.3 Adverse reactions -- 8.4 Warning and precautions -- 8.4.1 Infections -- 8.4.2 Diarrhea or colitis -- 8.4.3 Cutaneous reactions -- 8.4.4 Pneumonitis -- 8.4.5 Hepatotoxicity -- 8.4.6 Neutropenia -- 8.4.7 Embryo-fetal toxicity -- 8.5 Use in specific population -- 8.5.1 Pregnancy -- 8.5.2 Breastfeeding -- 8.5.3 Pediatric use -- 8.5.4 Hepatic impairment -- 8.5.5 Renal impairment -- References -- Chapter Three: Regorafenib: A comprehensive drug profile -- 1 Description -- 1.1 Nomenclature -- 1.1.1 Systematic chemical names [1] -- 1.1.2 Nonproprietary names [1] -- 1.1.3 Proprietary names [1] -- 1.2 Formulae [1] -- 1.2.1 Empirical formula, molecular weight, CAS number -- 1.2.2 Structural formula [1] -- 1.2.3 Simplified molecular input line entry system (SMILES) [1] -- 1.2.4 The IUPAC international chemical identifier (InChI) [1] -- 1.3 Elemental analysis -- 1.4 Appearance [2] -- 2 Physical characteristics -- 2.1 Ionization constants -- 2.2 Solubility characteristics -- 2.3 Partition coefficients -- 2.4 Crystallographic properties -- 2.4.1 X-ray powder diffraction pattern -- 2.5 Thermal methods of analysis -- 2.5.1 Melting behavior -- 2.5.2 Differential scanning calorimetry (DSC) -- 2.6 Spectroscopic identification -- 2.6.1 UV/VIS spectroscopy -- 2.6.2 Vibrational spectroscopy -- 2.7 Nuclear magnetic resonance spectrometry -- 2.7.1 1H NMR spectrum -- 2.7.2 13C NMR spectrum -- 2.8 Mass spectrometry -- 3 Methods of preparation -- 4 Methods of analysis -- 4.1 Electrochemical methods of analysis -- 4.2 Spectrophotometric methods of analysis -- 4.3 Chromatographic methods of analysis -- 5 Pharmacology -- 5.1 Pharmacokinetics -- 5.1.1 Absorption -- 5.1.2 Distribution -- 5.1.3 Elimination -- 5.1.4 Metabolism. 
505 8 |a 5.1.5 Excretion -- 5.2 Pharmacological effects -- 5.3 Drug-drug interactions -- References -- Chapter Four: Ponatinib: A comprehensive drug profile -- 1 General information -- 1.1 Nomenclature -- 1.1.1 Systematic chemical names -- 1.1.1.1 Ponatinib base [1] -- 1.1.1.2 Ponatinib hydrochloride -- 1.1.2 Non-proprietary names (generic names) -- 1.1.3 Proprietary names (brand Names) -- 1.2 Formulae -- 1.2.1 Empirical formula, molecular weight, and CAS number -- 1.2.2 Structural formula -- 1.3 Elemental analysis -- 1.4 Appearance -- 2 Physical characteristics -- 2.1 Dissociation constants -- 2.2 Solubility characteristics -- 2.3 Partition coefficients -- 2.4 Crystallographic properties -- 2.4.1 Single crystal structure [9] -- 2.4.2 X-ray powder diffraction pattern -- 2.5 Thermal gravimetric analysis (TGA) -- 2.6 Spectroscopy -- 2.6.1 Ultraviolet spectroscopy -- 2.6.2 Nuclear magnetic resonance spectrometry -- 2.6.2.1 1H NMR spectrum -- 2.6.2.2 13C NMR spectrum -- 2.6.3 Infrared spectroscopy -- 2.7 Mass spectrometry -- 3 Uses and applications -- 4 Stability -- 5 Preparation of ponatinib -- 6 Impurities -- 7 Reported methods of analysis -- 7.1 Electrochemical approach -- 7.2 Spectroscopic methods of analysis -- 7.2.1 Spectrofluorimetric method -- 7.2.2 Stimulated raman scattering (SRS) microscopy -- 7.3 Chromatographic methods of analysis -- 7.4 Immunoassay -- 8 Clinical pharmacology -- 8.1 Mechanism of action -- 8.2 Pharmacokinetics -- 8.2.1 Absorption -- 8.2.2 Distribution -- 8.2.3 Metabolism -- 8.2.4 Excretion -- 8.2.5 Special populations -- 8.3 Pharmacodynamics -- 8.4 Dosage -- 8.5 Adverse effects -- 8.6 Drug interactions -- References -- Chapter Five: Avanafil: A comprehensive drug profile -- 1 Description -- 1.1 Nomenclature -- 1.1.1 IUPAC names -- 1.1.1.1 Avanafil -- 1.1.1.2 Avanafil dibenzenesulfonate -- 1.1.2 Nonproprietary name. 
505 8 |a 1.1.3 Proprietary names -- 1.2 Formulae -- 1.2.1 Empirical formula, molecular weight, and CAS no -- 1.2.2 Structural formula -- 1.3 Elemental analysis -- 2 Methods of preparation of avanafil -- 3 Physical characteristics -- 3.1 Physical appearance -- 3.2 Specific rotation -- 3.3 Melting point -- 3.4 Dissociation constant -- 3.5 Solubility and partition coefficient -- 3.6 Stability -- 3.7 Crystallographic properties -- 3.8 Thermal analysis -- 3.9 Spectroscopy -- 3.9.1 UV/Vis spectroscopy -- 3.9.2 Spectrofluorimetric method -- 3.9.3 Infrared spectroscopy -- 3.9.3.1 Mass spectroscopy -- 3.9.4 NMR spectroscopy -- 3.9.4.1 1H NMR spectroscopy -- 3.9.5 13C NMR spectroscopy -- 4 Methods of analysis -- 4.1 Compendial method -- 4.2 Reported methods of analysis -- 4.2.1 Electrochemical methods -- 4.2.2 Spectroscopic methods -- 4.2.2.1 Colorimetric method -- 4.2.2.2 Spectrophotometry method -- 4.2.2.3 Spectrofluorimetric method -- 4.2.3 Capillary electrophoresis -- 4.2.4 Chromatography -- 4.2.4.1 High-performance thin-layer chromatography (HPTLC) methods -- 4.2.4.2 High-performance liquid chromatography methods -- 4.2.4.3 Liquid chromatography-tandem mass spectrometric methods (LC/MS) -- 4.2.4.4 Gas chromatography-mass spectrometry (GC/MS) -- 5 Stability -- 6 Clinical pharmacology of avanafil -- 6.1 Mechanism of action -- 6.2 Pharmacokinetics -- 6.2.1 Absorption -- 6.2.2 Distribution -- 6.2.3 Metabolism -- 6.2.4 Elimination -- 6.2.5 Special populations -- 6.3 Dosage and administration -- 6.4 Drug interactions -- 6.5 Adverse effects -- 6.6 Effects on the body -- References -- Chapter Six: Regulation and standardization of herbal drugs: Current status, limitation, challenge's and future prospective -- 1 Introduction -- 2 Regulation of herbal drugs -- 2.1 US Food and Drug Administration (FDA) -- 2.2 European Medicines Agency (EMA). 
505 8 |a 2.3 Pharmaceutical and Medical Devices Agency (PMDA) of Japan -- 2.4 Ministry of Health and Welfare Taiwan, Republic of China -- 2.5 Chinese Medicine Regulatory Office, Department of Health, The Government of Hong Kong Special Administrative Region -- 2.6 Indonesian National Agency of Drug and Food Control (BPOM-RI) -- 2.7 Summary and discussions -- 3 Standardization of herbal drugs: current criteria and limitations -- 3.1 Sampling and identification -- 3.2 Quantitative determination -- 3.3 Specific tests -- 3.4 Microbial quality tests -- 3.5 Summary and discussion -- 4 Challenges and future perspective of HD standardization methods -- 4.1 Qualitative method (identification) -- 4.2 Quantitative analysis and limit tests -- 5 Summary and recommendations -- Acknowledgments -- References -- Cumulative index -- Back Cover. 
588 |a Description based on print version record. 
504 |a Includes bibliographical references. 
650 0 |a Pharmaceutical chemistry. 
650 2 |a Chemistry, Pharmaceutical 
650 6 |a Chimie pharmaceutique. 
655 7 |a Electronic books.  |2 local 
700 1 |a Al-Majed, Abdulrahman,  |e editor. 
710 2 |a ScienceDirect (Online service) 
830 0 |a Profiles of drug substances, excipients, and related methodology ;  |v Volume 49. 
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