Drug selectivity : an evolving concept in medicinal chemistry /

Bibliographic Details
Other Authors: Handler, Norbert (Editor), Buschmann, Helmut (Editor)
Format: eBook
Language:English
Published: Weinheim, Germany : Wiley-VCH, [2018]
Series:Methods and principles in medicinal chemistry ; v. 72.
Subjects:
Online Access:Connect to the full text of this electronic book
Table of Contents:
  • Introduction. Polypharmacology in Drug Discovery / Oscar Méndez-Lucio, J Jesús Naveja, Hugo Vite-Caritino, Fernando D Prieto-Martínez, José L Medina-Franco
  • Selectivity of Marketed Drugs. Kinase Inhibitors / Peng Wu, Michael Givskov, Thomas E Nielsen
  • Repositioning of Drug
  • New Indications for Marketed Drugs / Ren Kong, Stephen T Wong
  • Discovery Technologies for Drug Repurposing / Naiem T Issa, Stephen W Byers, Sivanesan Dakshanamurthy
  • Unselective Drugs in Drug Discovery. Personalized Medicine / Christian Noe, Volker Baumann
  • Drug Discovery Strategies for the Generation of Multitarget Ligands against Neglected Tropical Diseases / Annachiara Gandini, Federica Prati, Elisa Uliassi, Maria L Bolognesi
  • Designing Approaches to Multitarget Drugs / Luca Costantino, Daniela Barlocco
  • The Linker Approach / Daniel Merk, Manfred Schubert-Zsilavecz
  • Merged Multiple Ligands / Hongming Chen, Udo Bauer, Ola Engkvist
  • Pharmacophore Generation for Multiple Ligands / Norbert Handler
  • Cellular Assays / Ye Fang
  • Therapeutic Areas for Designed Multiple Ligands. Developing Serotonergic Antidepressants Acting on More Than the Serotonin Transporter / Gerard J Marek
  • Multiple Ligands Targeting the Angiotensin System for Hypertension / Agustin Casimiro-Garcia
  • Multiple Peroxisome Proliferator-Activated Receptor-Based Ligands / Dmytro Kukhtar, Miquel Mulero, Raul Beltrán-Debón, Cristina Valls, Gerard Pujadas, Santiago Garcia-Vallve
  • Antibiotics / Jean-Philippe Surivet, Philippe Panchaud
  • Multiple Ligands in Neurodegenerative Diseases / Julien Lalut, Christophe Rochais, Patrick Dallemagne.