Optimizing the "drug-like" properties of leads in drug discovery /

Bibliographic Details
Other Authors: Borchardt, Ronald T.
Format: Book
Language:English
Published: New York, NY : Springer, [2006]
Series:Biotechnology (Arlington, Va.)
Subjects:

MARC

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245 0 0 |a Optimizing the "drug-like" properties of leads in drug discovery /  |c Ronald T. Borchardt [and others], editors. 
264 1 |a New York, NY :  |b Springer,  |c [2006] 
264 4 |c ©2006 
300 |a x, 512 pages :  |b illustrations (some color) ;  |c 27 cm +  |e 1 CD-ROM. 
336 |a text  |2 rdacontent  |b txt 
337 |a unmediated  |2 rdamedia 
338 |a volume  |2 rdacarrier  |b nc 
490 1 |a Biotechnology: pharmaceutical aspects 
500 |a "This book is based on proceedings from a worshop that took place in Parsippany, NJ on September 19-22, 2004." -- p. vii. 
504 |a Includes bibliographical references and index. 
505 0 |a Strategic use of preclinical pharmacokinetic studies and In Vitro models in optimizing ADME properties of lead compounds -- Role of mechanistic transport studies in lead optimization -- Metabolic activation-role in toxicity and idiosyncratic reactions -- Case history - use of ADME studies for optimization of drug candidates -- Solubility, solubilization and dissolution in drug delivery during lead optimization -- Lipid-based systems, drug exposure and lead optimization -- Biopharmaceutics modeling and the role of dose and formulation on oral exposure -- Application of physicochemical data to support lead optimization by discovery teams -- Computational models supporting lead optimization in drug discovery -- Prodrug strategies for improving drug-like properties -- The application of multivariate data analysis to compound property optimization -- Case history : toxicology biomarker development using toxicogenomics -- Predicting idiosyncratic drug reactions -- Elementary predictive toxicology for advanced applications -- The application of PK/PD modeling and simulations during lead optimization -- Early preclinical evaluation of brain exposure in support of hit identification and lead optimization -- Optimizing biomarker development for clinical studies at the lead optimization stage of drug development -- The relevance of transporters in determining drug disposition 
650 0 |a Drugs  |x Design. 
650 0 |a Drug development. 
650 0 |a Pharmaceutical chemistry. 
650 2 |a Drug Design. 
650 2 |a Chemistry, Pharmaceutical. 
700 1 |a Borchardt, Ronald T. 
830 0 |a Biotechnology (Arlington, Va.) 
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