Chemoinformatics : concepts, methods, and tools for drug discovery /

Bibliographic Details
Other Authors: Bajorath, Jürgen
Format: Book
Language:English
Published: Totowa, N.J. : Humana Press, [2004]
Series:Methods in molecular biology (Clifton, N.J.) ; v. 275.
Subjects:
Table of Contents:
  • Molecular similarity measures
  • Evaluation of molecular similarity and molecular diversity methods using biological activity data
  • A web-based chemoinformatics system for drug discovery
  • Application of chemoinformatics to high throughput screening : practical considerations
  • Strategies for the identification and generation of informative compound sets
  • Methods for applying the quantitative structure-activity relationship paradigm
  • 3D-LogP : an alignment-freee 3D description of local lipophilicity for QSAR studies
  • Derivation and applications of molecular descriptors based on approximate surface area
  • Cell-based partitioning in binary-transformed chemical descriptor spaces
  • Comparison of methods based on diversity and similarity for molecule selection and the analysis of drug discovery data
  • Using recursive partitioning analysis to evaluate compound selection methods
  • Designing combinatorial libraries optimized on multiple objectives
  • Approaches to target class combinatorial library design
  • Simulated annealing : an effective stochastic optimization approach to computational library design
  • Genetic algorithms for classification of olfactory stimulants
  • How to describe chirality and conformational flexibility
  • Novel scoring methods in virtual ligand screening
  • Prediction of drug-like molecular properties : modeling cytochrome P450 interactions