Combinatorial library : methods and protocols /

Bibliographic Details
Other Authors: English, Lisa Bellavance
Format: Book
Language:English
Published: Totowa, N.J. : Humana Press, [2002]
Series:Methods in molecular biology (Clifton, N.J.) ; v. 201.
Subjects:
Table of Contents:
  • Pt. I. Library synthesis and quality control
  • Using a noncovalent protection strategy to enhance solid-phase synthesis
  • Quality control of solid-phase synthesis by mass spectrometry
  • Preparation of encoded combinatorial libraries for drug discovery
  • Simple tools for manual parallel solid phase synthesis
  • Cleavage of compounds from solid phase by gaseous reagents
  • Synthesis of DNA-binding polyamides : robust solid-phase methods for coupling heterocyclic aromatic amino acids
  • The preparation of phenyl-stilbene derivatives using the safety catch linker
  • Host-guest chemistry : combinatorial receptors
  • Automated structure verification of small molecules libraries using 1D and 2D NMR techniques
  • Rapid liquid-phase combinatorial synthesis of heterocyclic libraries
  • Soluble polymer-supported methods for combinatorial and organic synthesis
  • Analytical methods for optimization and quality control of combinatorial synthesis
  • Pt. II. Library purification and screening
  • Resolving racemic mixtures using parallel combinatorial libraries
  • Ligand libraries for the extraction of metal ions : dynamic combinatorial and high-throughout screening methods
  • Automated liquid-liquid extraction and ion-exchange solid-phase extraction for initial purification
  • On-bead and solution screening approaches for genomically derived targets : discovery of surrogate ligands and substrates using combinatorial chemistry libraries
  • Pt. III. Computational library design
  • Design of virtual combinatorial libraries
  • Approaches to library design for combinatorial chemistry
  • Reagent-based and product-based computational strategies in library design
  • Designing combinatorial libraries for efficient screening
  • Application of neural networks to large dataset QSAR, virtual screening, and library design